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|  | ANNEX A-1: Merger Agreement |  |  |  |  |  |  |  | 
|  | ANNEX A-2: Merger Agreement Amendment |  |  |  |  |  |  |  | 
|  | ANNEX B: Form of CVR Agreement |  |  |  |  |  |  |  | 
|  | ANNEX C: Opinion of Locust Walk Securities, LLC |  |  |  |  |  |  |  | 
|  | ANNEX D: Opinion of Kroll, LLC |  |  |  |  |  |  |  | 
|  | ANNEX E: Royalty Agreement |  |  |  |  |  |  |  | 
|  | ANNEX F: Support Agreement |  |  |  |  |  |  |  | 
|  | ANNEX G: Form of Transition Services Agreement |  |  |  |  |  |  |  | 
|  | ANNEX H: Warrant Amendment |  |  |  |  |  |  |  | 
| 
                Company 
               |  |  | 
                Stage of 
                 Development |  |  | 
                Stock 
                 Price(1) |  |  | 
                Enterprise 
                 Value ($M)(1) |  |  | 
                Peak 
                 Sales(2) ($M) |  |  | 
                Enterprise 
                 Value / Peak Sales(2) |  |  | 
                5-Year 
                 Projected Sales (2029)(3) |  |  | 
                Enterprise 
                 Value / 5-Year Sales (2029)(3) |  | ||||||||||||||||||
| 
                Adaptimmune Therapeutics 
               |  |  | 
                Approved 
               |  |  |  | $ | 0.54 |  |  |  |  | $ | 2 |  |  |  |  | $ | 397 |  |  |  |  |  | 0.00x |  |  |  |  | $ | 137 |  |  |  |  |  | 0.0x |  |  | 
| 
                ADC Therapeutics 
               |  |  | 
                Approved 
               |  |  |  | $ | 1.99 |  |  |  |  | $ | 32 |  |  |  |  | $ | 851 |  |  |  |  |  | 0.04x |  |  |  |  | $ | 247 |  |  |  |  |  | 0.1x |  |  | 
| 
                Iteos Therapeutics 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 7.68 |  |  |  |  | $ | 208 |  |  |  |  | $ | 1,277 |  |  |  |  |  | 0.16x |  |  |  |  | $ | 41 |  |  |  |  |  | 5.1x |  |  | 
| 
                Olema Pharmaceuticals 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 5.83 |  |  |  |  | $ | 37 |  |  |  |  | $ | 4,725 |  |  |  |  |  | 0.01x |  |  |  |  | $ | 495 |  |  |  |  |  | 0.1x |  |  | 
| 
                Aura Biosciences 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 8.22 |  |  |  |  | $ | 236 |  |  |  |  | $ | 1,286 |  |  |  |  |  | 0.18x |  |  |  |  | $ | 288 |  |  |  |  |  | 0.8x |  |  | 
| 
                Candel Therapeutics 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 8.68 |  |  |  |  | $ | 366 |  |  |  |  | $ | 818 |  |  |  |  |  | 0.45x |  |  |  |  | $ | 261 |  |  |  |  |  | 1.4x |  |  | 
| 
                Celcuity 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 13.09 |  |  |  |  | $ | 726 |  |  |  |  | $ | 1,718 |  |  |  |  |  | 0.42x |  |  |  |  | $ | 598 |  |  |  |  |  | 1.2x |  |  | 
| 
                Compass Therapeutics 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 1.45 |  |  |  |  | $ | 64 |  |  |  |  | $ | 1,114 |  |  |  |  |  | 0.06x |  |  |  |  | $ | 364 |  |  |  |  |  | 0.2x |  |  | 
| 
                Erasca 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 2.51 |  |  |  |  | $ | 391 |  |  |  |  | $ | 4,336 |  |  |  |  |  | 0.09x |  |  |  |  | $ | 199 |  |  |  |  |  | 2.0x |  |  | 
| 
                75th Percentile 
               |  |  |  |  |  |  |  |  |  |  |  |  | $ | 366 |  |  |  |  | $ | 1,718 |  |  |  |  |  | 0.18x |  |  |  |  | $ | 364 |  |  |  |  |  | 1.4x |  |  | 
| 
                Median 
               |  |  |  |  |  |  |  |  |  |  |  |  | $ | 208 |  |  |  |  | $ | 1,277 |  |  |  |  |  | 0.09x |  |  |  |  | $ | 261 |  |  |  |  |  | 0.8x |  |  | 
| 
                25th Percentile 
               |  |  |  |  |  |  |  |  |  |  |  |  | $ | 37 |  |  |  |  | $ | 851 |  |  |  |  |  | 0.04x |  |  |  |  | $ | 199 |  |  |  |  |  | 0.1x |  |  | 
| 
                Metric 
               |  |  | 
                Metric Value 
               |  |  |  |  |  | 
                Enterprise 
                 Value / Peak Sales Multiple |  |  | 
                Implied 
                 Enterprise Value ($M) |  | |||||||||
| 
                The Company Peak Sales ($M) 
               |  |  |  | $ | 649(2) |  |  |  | 
                75th Percentile 
               |  |  |  |  | 0.18x |  |  |  |  | $ | 119 |  |  | 
|  |  |  |  |  |  |  |  |  | 
                Median 
               |  |  |  |  | 0.09x |  |  |  |  | $ | 58 |  |  | 
|  |  |  |  |  |  |  |  |  | 
                25th Percentile 
               |  |  |  |  | 0.04x |  |  |  |  | $ | 25 |  |  | 
| 
                The Company 5-Year Sales ($M) 
               |  |  |  | $ | 237(3) |  |  |  | 
                75th Percentile 
               |  |  |  |  | 1.4x |  |  |  |  | $ | 332 |  |  | 
|  |  |  |  |  |  |  |  |  | 
                Median 
               |  |  |  |  | 0.8x |  |  |  |  | $ | 190 |  |  | 
|  |  |  |  |  |  |  |  |  | 
                25th Percentile 
               |  |  |  |  | 0.1x |  |  |  |  | $ | 24 |  |  | 
| 
                Date 
               |  |  | 
                Seller 
               |  |  | 
                Buyer 
               |  |  | 
                Stage of 
                 Development |  |  | 
                Deal 
                 Value ($M) |  |  | 
                Offer Price 
                 per Share |  |  | 
                30-Day 
                 VWAP(1) |  |  | 
                Equity 
                 Premium(2) |  | ||||||||||||
| 
                Apr-24 
               |  |  | 
                Deciphera Pharmaceuticals 
               |  |  | 
                Ono Pharmaceutical 
               |  |  | 
                Approved 
               |  |  |  | $ | 2,400 |  |  |  |  | $ | 25.60 |  |  |  |  | $ | 15.20 |  |  |  |  |  | 68% |  |  | 
| Mar-24 |  |  | 
                Fusian Pharmaceuticals 
               |  |  | 
                AstraZenenca 
               |  |  | 
                Phase 2 
               |  |  |  | $ | 2,000 |  |  |  |  | $ | 21.00 |  |  |  |  | $ | 11.40 |  |  |  |  |  | 84% |  |  | 
| 
                Jan-24 
               |  |  | 
                Harpoon Therapeutics 
               |  |  | 
                Merck 
               |  |  | 
                Phase 2 
               |  |  |  | $ | 680 |  |  |  |  | $ | 23.00 |  |  |  |  | $ | 10.71 |  |  |  |  |  | 115% |  |  | 
| 
                Jan-24 
               |  |  | 
                Ambrx 
               |  |  | 
                Johnson & Johnson 
               |  |  | 
                Phase 2 
               |  |  |  | $ | 2,000 |  |  |  |  | $ | 28.00 |  |  |  |  | $ | 13.03 |  |  |  |  |  | 115% |  |  | 
| 
                Dec-23 
               |  |  | 
                RayzeBio 
               |  |  | 
                BMS 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 4,100 |  |  |  |  | $ | 62.50 |  |  |  |  | $ | 25.80 |  |  |  |  |  | 142% |  |  | 
| 
                Oct-23 
               |  |  | 
                Mirati 
               |  |  | 
                BMS 
               |  |  | 
                Approved 
               |  |  |  | $ | 4,800 |  |  |  |  | $ | 58.00 |  |  |  |  | $ | 37.94 |  |  |  |  |  | 53% |  |  | 
| 
                Oct-23 
               |  |  | 
                Point Biopharma 
               |  |  | 
                Eli Lilly 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 1,400 |  |  |  |  | $ | 12.50 |  |  |  |  | $ | 7.44 |  |  |  |  |  | 68% |  |  | 
| 
                Oct-22 
               |  |  | 
                AVEO 
               |  |  | 
                LG Chem 
               |  |  | 
                Approved 
               |  |  |  | $ | 566 |  |  |  |  | $ | 15.00 |  |  |  |  | $ | 8.35 |  |  |  |  |  | 80% |  |  | 
| 
                Jun-22 
               |  |  | 
                F-Star 
               |  |  | 
                invoX Pharma 
               |  |  | 
                Phase 2 
               |  |  |  | $ | 161 |  |  |  |  | $ | 7.12 |  |  |  |  | $ | 3.13 |  |  |  |  |  | 128% |  |  | 
| 
                Jun-22 
               |  |  | 
                Turning Point 
               |  |  | 
                BMS 
               |  |  | 
                Phase 2 
               |  |  |  | $ | 4,100 |  |  |  |  | $ | 76.00 |  |  |  |  | $ | 31.29 |  |  |  |  |  | 143% |  |  | 
| 
                Apr-22 
               |  |  | 
                Checkmate Pharmaceuticals 
               |  |  | 
                Regeneron 
               |  |  | 
                Phase 2 
               |  |  |  | $ | 250 |  |  |  |  | $ | 10.50 |  |  |  |  | $ | 3.09 |  |  |  |  |  | 240% |  |  | 
| Mar-21 |  |  | 
                Five Prime 
               |  |  | 
                Amgen 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 1,900 |  |  |  |  | $ | 38.00 |  |  |  |  | $ | 18.87 |  |  |  |  |  | 101% |  |  | 
|  |  |  | 
                Equity Premium 
               |  |  |  |  |  |  |  |  |  |  |  |  |  |  | 
                75th
                 Percentile 
               |  |  | 
                Median 
               |  |  | 
                25th
                 Percentile 
               |  | |||||||||
|  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  | 
                139%
               |  |  | 
                108%
               |  |  | 
                71%
               |  | |||||||||
| 
                Date 
               |  |  | 
                Seller 
               |  |  | 
                Buyer 
               |  |  | 
                Stage of 
                 Development |  |  | 
                Deal 
                 Value ($M) |  |  | 
                Offer Price 
                 per Share |  |  | 
                30-Day 
                 VWAP(1) |  |  | 
                Equity 
                 Premium(2) |  | ||||||||||||
| 
                Oct-24 
               |  |  | 
                Longboard Pharmaceuticals 
               |  |  | 
                Lundbeck 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 2,500 |  |  |  |  | $ | 60 |  |  |  |  | $ | 34.52 |  |  |  |  |  | 74% |  |  | 
| 
                Aug-24 
               |  |  | 
                Revance Therapeutics 
               |  |  | 
                Crown Laboratories 
               |  |  | 
                Approved 
               |  |  |  | $ | 924 |  |  |  |  | $ | 6.66 |  |  |  |  | $ | 3.38 |  |  |  |  |  | 97% |  |  | 
| 
                Aug-24 
               |  |  | 
                G1 Therapeutics 
               |  |  | 
                Pharmacosmos 
               |  |  | 
                Approved 
               |  |  |  | $ | 405 |  |  |  |  | $ | 7.15 |  |  |  |  | $ | 3.07 |  |  |  |  |  | 133% |  |  | 
| 
                Jun-24 
               |  |  | 
                Alimera Sciences 
               |  |  | 
                ANI Pharmaceuticals 
               |  |  | 
                Approved 
               |  |  |  | $ | 381 |  |  |  |  | $ | 5.50 |  |  |  |  | $ | 3.05 |  |  |  |  |  | 80% |  |  | 
| 
                May-24 
               |  |  | 
                Calliditas Therapeutics 
               |  |  | 
                Asahi Kasei 
               |  |  | 
                Approved 
               |  |  |  | $ | 1,116(3) |  |  |  |  | $ | 39.09(3) |  |  |  |  | $ | 20.38(3) |  |  |  |  |  | 92% |  |  | 
| 
                Apr-24 
               |  |  | 
                Deciphera Pharmaceuticals 
               |  |  | 
                Ono Pharmaceuticals 
               |  |  | 
                Approved 
               |  |  |  | $ | 2,400 |  |  |  |  | $ | 25.60 |  |  |  |  | $ | 15.20 |  |  |  |  |  | 68% |  |  | 
| 
                Feb-24 
               |  |  | 
                CymaBay Therapeutics 
               |  |  | 
                Gilead Sciences 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 4,300 |  |  |  |  | $ | 32.50 |  |  |  |  | $ | 23.80 |  |  |  |  |  | 37% |  |  | 
| 
                Feb-24 
               |  |  | 
                MorphaSys 
               |  |  | 
                Novartis 
               |  |  | 
                Phase 3 
               |  |  |  | € | 2,700 |  |  |  |  | € | 68.00 |  |  |  |  | € | 34.88 |  |  |  |  |  | 95% |  |  | 
|  |  |  | 
                Equity Premium 
               |  |  |  |  |  |  |  |  |  |  |  |  |  |  | 
                75th
                 Percentile 
               |  |  | 
                Median 
               |  |  | 
                25th
                 Percentile 
               |  | |||||||||
|  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  | 
                96% 
               |  |  | 
                86% 
               |  |  | 
                73%
               |  | |||||||||
| 
                Date 
               |  |  | 
                Seller 
               |  |  | 
                Buyer 
               |  |  | 
                Stage of 
                 Development |  |  | 
                Deal 
                 Value ($M) |  |  | 
                Offer Price 
                 per Share |  |  | 
                30-Day 
                 VWAP(1) |  |  | 
                Equity 
                 Premium(2) |  | ||||||||||||
| 
                Aug-24 
               |  |  | 
                Revance Therapeutics 
               |  |  | 
                Crown Laboratories 
               |  |  | 
                Approved 
               |  |  |  | $ | 924 |  |  |  |  | $ | 6.66 |  |  |  |  | $ | 3.38 |  |  |  |  |  | 97% |  |  | 
| 
                Aug-24 
               |  |  | 
                G1 Therapeutics 
               |  |  | 
                Pharmacosmos 
               |  |  | 
                Approved 
               |  |  |  | $ | 405 |  |  |  |  | $ | 7.15 |  |  |  |  | $ | 3.07 |  |  |  |  |  | 133% |  |  | 
| 
                Jun-24 
               |  |  | 
                Alimera Sciences 
               |  |  | 
                ANI Pharmaceuticals 
               |  |  | 
                Approved 
               |  |  |  | $ | 381 |  |  |  |  | $ | 5.50 |  |  |  |  | $ | 3.05 |  |  |  |  |  | 80% |  |  | 
| 
                May-24 
               |  |  | 
                Calliditas Therapeutics 
               |  |  | 
                Asahi Kasei 
               |  |  | 
                Approved 
               |  |  |  | $ | 1,116(3) |  |  |  |  | $ | 39.09(3) |  |  |  |  | $ | 20.38(3) |  |  |  |  |  | 92% |  |  | 
| 
                Apr-24 
               |  |  | 
                Deciphera Pharmaceuticals 
               |  |  | 
                Ono Pharmaceuticals 
               |  |  | 
                Approved 
               |  |  |  | $ | 2,400 |  |  |  |  | $ | 25.60 |  |  |  |  | $ | 15.20 |  |  |  |  |  | 68% |  |  | 
|  |  |  | 
                Equity Premium 
               |  |  |  |  |  |  |  |  | 
                75th
                 Percentile 
               |  |  | 
                Median 
               |  |  | 
                25th
                 Percentile
               |  |  |  |  |  |  |  | |||||||||
|  |  |  |  |  |  |  |  |  |  |  |  | 
                97% 
               |  |  | 
                86% 
               |  |  | 
                74%
               |  |  |  |  |  |  |  | |||||||||
| 
                Date 
               |  |  | 
                Seller 
               |  |  | 
                Buyer 
               |  |  | 
                Stage of 
                 Development |  |  | 
                Deal 
                 Value ($M) |  |  | 
                Offer Price 
                 per Share |  |  | 
                30-Day 
                 VWAP(1) |  |  | 
                Equity 
                 Premium(2) |  | ||||||||||||
| 
                Jun-23 
               |  |  | 
                Paratek Pharmaceuticals 
               |  |  | 
                Gurnet Point Capital / 
                 Novo Holdings |  |  | 
                Approved 
               |  |  |  | $ | 331 |  |  |  |  | $ | 2.15 |  |  |  |  | $ | 1.77 |  |  |  |  |  | 21% |  |  | 
| 
                Jan-23 
               |  |  | 
                Concert Pharmaceuticals 
               |  |  | 
                Sun Pharma 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 576 |  |  |  |  | $ | 8.00 |  |  |  |  | $ | 5.98 |  |  |  |  |  | 34% |  |  | 
| 
                Nov-22 
               |  |  | 
                Opiant Pharmaceuticals 
               |  |  | 
                Indivior 
               |  |  | 
                Phase 3 
               |  |  |  | $ | 145 |  |  |  |  | $ | 20.00 |  |  |  |  | $ | 10.12 |  |  |  |  |  | 98% |  |  | 
| 
                Nov-22 
               |  |  | 
                Oyster Point Pharma 
               |  |  | 
                Viatris 
               |  |  | 
                Approved 
               |  |  |  | $ | 415 |  |  |  |  | $ | 11.00 |  |  |  |  | $ | 7.14 |  |  |  |  |  | 54% |  |  | 
| 
                Jun-22 
               |  |  | 
                Radius Health 
               |  |  | 
                Gurnet Point Capital / 
                 Patient Square Capital |  |  | 
                Approved 
               |  |  |  | $ | 497 |  |  |  |  | $ | 10.00 |  |  |  |  | $ | 6.94 |  |  |  |  |  | 44% |  |  | 
|  |  |  | 
                Equity Premium 
               |  |  |  |  |  |  |  |  | 
                75th
                 Percentile 
               |  |  | 
                Median 
               |  |  | 
                25th
                 Percentile 
               |  |  |  |  |  |  |  | |||||||||
|  |  |  |  |  |  |  |  |  |  |  |  | 
                54% 
               |  |  | 
                44% 
               |  |  | 
                34% 
               |  |  |  |  |  |  |  | |||||||||
|  |  |  | 
                2025 
               |  |  | 
                2026 
               |  |  | 
                2027 
               |  |  | 
                2028 
               |  |  | 
                2029 
               |  | |||||||||||||||
| 
                Net Revenue(1)
               |  |  |  | $ | 17.2 |  |  |  |  | $ | 113.0 |  |  |  |  | $ | 277.6 |  |  |  |  | $ | 417.1 |  |  |  |  | $ | 479.6 |  |  | 
|  |  |  | 
                2024 
               |  |  | 
                2025 
               |  |  | 
                2026 
               |  |  | 
                2027 
               |  |  | 
                2028 
               |  |  | 
                2029 
               |  |  | 
                2030 
               |  |  | 
                2031 
               |  |  | 
                2032 
               |  |  | 
                2033 
               |  |  | 
                2034 
               |  |  | 
                2035 
               |  |  | 
                2036 
               |  |  | 
                2037 
               |  |  | 
                2038 
               |  | |||||||||||||||||||||||||||||||||||||||||||||
| 
                Risk-Adjusted Net 
                 Revenue(1) |  |  |  |  | — |  |  |  |  | $ | 1.9 |  |  |  |  | $ | 43.4 |  |  |  |  | $ | 142.3 |  |  |  |  | $ | 227.6 |  |  |  |  | $ | 195.7 |  |  |  |  | $ | 209.7 |  |  |  |  | $ | 217.0 |  |  |  |  | $ | 224.6 |  |  |  |  | $ | 232.5 |  |  |  |  | $ | 240.6 |  |  |  |  | $ | 249.1 |  |  |  |  | $ | 257.8 |  |  |  |  | $ | 266.8 |  |  |  |  | $ | 276.1 |  |  | 
| 
                Risk-Adjusted 
                 EBIT(2) |  |  |  |  | — |  |  |  |  | $ | (46.1) |  |  |  |  | $ | (3.9) |  |  |  |  | $ | 81.5 |  |  |  |  | $ | 133.0 |  |  |  |  | $ | 94.3 |  |  |  |  | $ | 98.2 |  |  |  |  | $ | 99.5 |  |  |  |  | $ | 101.4 |  |  |  |  | $ | 103.0 |  |  |  |  | $ | 106.4 |  |  |  |  | $ | 110.3 |  |  |  |  | $ | 114.7 |  |  |  |  | $ | 119.2 |  |  |  |  | $ | 123.8 |  |  | 
| 
                Risk-Adjusted Unlevered Free Cash Flow(3)
               |  |  |  |  | — |  |  |  |  | $ | (63.4) |  |  |  |  | $ | (27.5) |  |  |  |  | $ | 49.4 |  |  |  |  | $ | 110.7 |  |  |  |  | $ | 94.2 |  |  |  |  | $ | 87.6 |  |  |  |  | $ | 78.6 |  |  |  |  | $ | 71.2 |  |  |  |  | $ | 72.3 |  |  |  |  | $ | 74.5 |  |  |  |  | $ | 77.3 |  |  |  |  | $ | 80.3 |  |  |  |  | $ | 83.5 |  |  |  |  | $ | 86.7 |  |  | 
|  |  |  | 
                2024 
               |  |  | 
                2025 
               |  |  | 
                2026 
               |  |  | 
                2027 
               |  |  | 
                2028 
               |  |  | 
                2029 
               |  |  | 
                2030 
               |  |  | 
                2031 
               |  |  | 
                2032 
               |  |  | 
                2033 
               |  |  | 
                2034 
               |  |  | 
                2035 
               |  |  | 
                2036 
               |  |  | 
                2037 
               |  |  | 
                2038 
               |  | |||||||||||||||||||||||||||||||||||||||||||||
| 
                Risk-Adjusted Net Revenue(1)
               |  |  |  |  | — |  |  |  |  | $ | 1.9 |  |  |  |  | $ | 43.6 |  |  |  |  | $ | 147.1 |  |  |  |  | $ | 252.7 |  |  |  |  | $ | 254.1 |  |  |  |  | $ | 286.2 |  |  |  |  | $ | 286.9 |  |  |  |  | $ | 298.8 |  |  |  |  | $ | 309.2 |  |  |  |  | $ | 320.0 |  |  |  |  | $ | 331.2 |  |  |  |  | $ | 342.8 |  |  |  |  | $ | 354.8 |  |  |  |  | $ | 367.3 |  |  | 
| 
                Risk-Adjusted 
                 EBIT(2) |  |  |  |  | — |  |  |  |  | $ | (46.1) |  |  |  |  | $ | (4.6) |  |  |  |  | $ | 80.4 |  |  |  |  | $ | 140.7 |  |  |  |  | $ | 105.2 |  |  |  |  | $ | 112.6 |  |  |  |  | $ | 112.7 |  |  |  |  | $ | 115.4 |  |  |  |  | $ | 109.9 |  |  |  |  | $ | 119.7 |  |  |  |  | $ | 124.2 |  |  |  |  | $ | 129.0 |  |  |  |  | $ | 134.0 |  |  |  |  | $ | 139.2 |  |  | 
| 
                Risk-Adjusted 
                 Unlevered Free Cash Flow(3) |  |  |  |  | — |  |  |  |  | $ | (63.4) |  |  |  |  | $ | (28.3) |  |  |  |  | $ | 47.3 |  |  |  |  | $ | 112.8 |  |  |  |  | $ | 95.5 |  |  |  |  | $ | 94.0 |  |  |  |  | $ | 92.6 |  |  |  |  | $ | 80.7 |  |  |  |  | $ | 76.9 |  |  |  |  | $ | 83.8 |  |  |  |  | $ | 86.9 |  |  |  |  | $ | 90.3 |  |  |  |  | $ | 93.8 |  |  |  |  | $ | 97.4 |  |  | 
|  |  |  | 
                2024 
               |  |  | 
                2025 
               |  |  | 
                2026 
               |  |  | 
                2027 
               |  |  | 
                2028 
               |  |  | 
                2029 
               |  |  | 
                2030 
               |  |  | 
                2031 
               |  |  | 
                2032 
               |  |  | 
                2033 
               |  |  | 
                2034 
               |  |  | 
                2035 
               |  |  | 
                2036 
               |  |  | 
                2037 
               |  |  | 
                2038 
               |  | |||||||||||||||||||||||||||||||||||||||||||||
| 
                Risk-Adjusted Net Revenue(1)
               |  |  |  |  | — |  |  |  |  | $ | 1.8 |  |  |  |  | $ | 41.2 |  |  |  |  | $ | 135.2 |  |  |  |  | $ | 216.3 |  |  |  |  | $ | 185.9 |  |  |  |  | $ | 199.2 |  |  |  |  | $ | 206.2 |  |  |  |  | $ | 213.4 |  |  |  |  | $ | 220.9 |  |  |  |  | $ | 228.6 |  |  |  |  | $ | 236.6 |  |  |  |  | $ | 244.9 |  |  |  |  | $ | 253.5 |  |  |  |  | $ | 262.3 |  |  | 
| 
                Risk-Adjusted EBIT(2)
               |  |  |  | $ | (27.8) |  |  |  |  | $ | (43.8) |  |  |  |  | $ | (3.8) |  |  |  |  | $ | 80.4 |  |  |  |  | $ | 158.1 |  |  |  |  | $ | 130.2 |  |  |  |  | $ | 137.7 |  |  |  |  | $ | 140.0 |  |  |  |  | $ | 143.5 |  |  |  |  | $ | 140.3 |  |  |  |  | $ | 150.8 |  |  |  |  | $ | 156.3 |  |  |  |  | $ | 162.3 |  |  |  |  | $ | 168.4 |  |  |  |  | $ | 174.8 |  |  | 
| 
                Risk-Adjusted Unlevered Free Cash Flow(3)
               |  |  |  | $ | (25.6) |  |  |  |  | $ | (43.2) |  |  |  |  | $ | (10.1) |  |  |  |  | $ | 60.4 |  |  |  |  | $ | 134.4 |  |  |  |  | $ | 127.7 |  |  |  |  | $ | 110.8 |  |  |  |  | $ | 101.3 |  |  |  |  | $ | 103.7 |  |  |  |  | $ | 101.4 |  |  |  |  | $ | 108.9 |  |  |  |  | $ | 112.9 |  |  |  |  | $ | 117.1 |  |  |  |  | $ | 121.6 |  |  |  |  | $ | 126.2 |  |  | 
|  |  |  | 
                2024 
               |  |  | 
                2025 
               |  |  | 
                2026 
               |  |  | 
                2027 
               |  |  | 
                2028 
               |  |  | 
                2029 
               |  |  | 
                2030 
               |  |  | 
                2031 
               |  |  | 
                2032 
               |  |  | 
                2033 
               |  |  | 
                2034 
               |  |  | 
                2035 
               |  |  | 
                2036 
               |  |  | 
                2037 
               |  |  | 
                2038 
               |  | |||||||||||||||||||||||||||||||||||||||||||||
| 
                Risk-Adjusted Net Revenue(1)
               |  |  |  |  | — |  |  |  |  | $ | 1.8 |  |  |  |  | $ | 41.4 |  |  |  |  | $ | 139.8 |  |  |  |  | $ | 240.1 |  |  |  |  | $ | 241.4 |  |  |  |  | $ | 271.9 |  |  |  |  | $ | 272.6 |  |  |  |  | $ | 283.8 |  |  |  |  | $ | 293.8 |  |  |  |  | $ | 304.0 |  |  |  |  | $ | 314.7 |  |  |  |  | $ | 325.7 |  |  |  |  | $ | 337.1 |  |  |  |  | $ | 348.9 |  |  | 
| 
                Risk-Adjusted EBIT(2)
               |  |  |  | $ | (27.8) |  |  |  |  | $ | (43.8) |  |  |  |  | $ | (3.8) |  |  |  |  | $ | 81.5 |  |  |  |  | $ | 163.3 |  |  |  |  | $ | 136.4 |  |  |  |  | $ | 145.9 |  |  |  |  | $ | 147.5 |  |  |  |  | $ | 151.4 |  |  |  |  | $ | 147.7 |  |  |  |  | $ | 158.5 |  |  |  |  | $ | 164.3 |  |  |  |  | $ | 170.5 |  |  |  |  | $ | 176.9 |  |  |  |  | $ | 183.6 |  |  | 
| 
                Risk-Adjusted Unlevered Free Cash Flow(3)
               |  |  |  | $ | (25.6) |  |  |  |  | $ | (43.2) |  |  |  |  | $ | (10.1) |  |  |  |  | $ | 60.3 |  |  |  |  | $ | 134.3 |  |  |  |  | $ | 125.0 |  |  |  |  | $ | 116.6 |  |  |  |  | $ | 107.7 |  |  |  |  | $ | 108.8 |  |  |  |  | $ | 106.4 |  |  |  |  | $ | 114.1 |  |  |  |  | $ | 118.2 |  |  |  |  | $ | 122.7 |  |  |  |  | $ | 127.3 |  |  |  |  | $ | 132.1 |  |  | 
|  |  |  | 
                Unvested Company Restricted Shares 
               |  | |||||||||||||||||||||
| 
                Name 
               |  |  | 
                Number of
                 Unvested Company Restricted Shares (#) |  |  | 
                Cash Amount
                 Payable in Respect of Unvested Company Restricted Shares ($) |  |  | 
                Number
                 of CVRs Issued in Respect of Unvested Company Restricted Shares (#) |  |  | 
                Maximum
                 Payment for CVRs Issued in Respect of Unvested Company Restricted Shares ($)(1) |  | ||||||||||||
| Executive Officers |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  | 
| 
                James F. Oliviero, III, President, Chief Executive Officer and Director 
               |  |  |  |  | 2,765,264 |  |  |  |  |  | 11,337,582 |  |  |  |  |  | 2,765,264 |  |  |  |  |  | 1,935,685 |  |  | 
| 
                William Garrett Gray, Chief Financial Officer, Corporate Secretary and Treasurer 
               |  |  |  |  | 913,425 |  |  |  |  |  | 3,745,043 |  |  |  |  |  | 913,425 |  |  |  |  |  | 639,398 |  |  | 
| Directors |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  | 
| 
                Michael S. Weiss, Chairman of the Checkpoint Board 
               |  |  |  |  | 104,295 |  |  |  |  |  | 427,610 |  |  |  |  |  | 104,295 |  |  |  |  |  | 73,007 |  |  | 
| 
                Christian Béchon, Director 
               |  |  |  |  | 104,295 |  |  |  |  |  | 427,610 |  |  |  |  |  | 104,295 |  |  |  |  |  | 73,007 |  |  | 
| 
                Neil Herskowitz, Director 
               |  |  |  |  | 104,295 |  |  |  |  |  | 427,610 |  |  |  |  |  | 104,295 |  |  |  |  |  | 73,007 |  |  | 
| 
                Lindsay A. Rosenwald, M.D. 
               |  |  |  |  | 104,295 |  |  |  |  |  | 427,610 |  |  |  |  |  | 104,295 |  |  |  |  |  | 73,007 |  |  | 
| 
                Barry Salzman, Director 
               |  |  |  |  | 104,295 |  |  |  |  |  | 427,610 |  |  |  |  |  | 104,295 |  |  |  |  |  | 73,007 |  |  | 
| 
                Amit Sharma, M.D., Director 
               |  |  |  |  | 82,051 |  |  |  |  |  | 336,409 |  |  |  |  |  | 82,051 |  |  |  |  |  | 57,436 |  |  | 
|  |  |  | 
                Unvested Company Restricted Shares 
               |  | |||||||||||||||||||||
| 
                Name 
               |  |  | 
                Number of
                 Unvested Company Restricted Shares (#) |  |  | 
                Cash Amount
                 Payable in Respect of Unvested Company Restricted Shares ($) |  |  | 
                Number
                 of CVRs Issued in Respect of Unvested Company Restricted Shares (#) |  |  | 
                Maximum
                 Payment for CVRs Issued in Respect of Unvested Company Restricted Shares ($)(1) |  | ||||||||||||
| 
                All of Checkpoint’s current directors and executive officers as a group (8 persons)
               |  |  |  |  | 4,282,215 |  |  |  |  |  | 17,557,084 |  |  |  |  |  | 4,282,215 |  |  |  |  |  | 2,997,554 |  |  | 
| 
                Name 
               |  |  | 
                Cash ($)(1)
               |  |  | 
                Equity ($)(2)
               |  |  | 
                Perquisites/ Benefits ($)(3) |  |  | 
                Other ($) 
               |  |  | 
                Total ($) 
               |  | |||||||||||||||
| 
                James F. Oliviero, III 
               |  |  |  |  | 1,759,920 |  |  |  |  |  | 13,273,267 |  |  |  |  |  | 35,000 |  |  |  |  |  | — |  |  |  |  |  | 15,068,187 |  |  | 
| 
                William Garrett Gray 
               |  |  |  |  | 828,375 |  |  |  |  |  | 4,384,440 |  |  |  |  |  | 35,000 |  |  |  |  |  | — |  |  |  |  |  | 5,247,815 |  |  | 
| 
                Name 
               |  |  | 
                Shares (#)(1)
               |  |  | 
                Shares ($) 
               |  |  | 
                Unvested 
                 Restricted Shares (#)(2)(3) |  |  | 
                Unvested 
                 Restricted Shares ($)(3) |  |  | 
                Total
                 ($) |  | |||||||||||||||
| Executive Officers |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  | 
| 
                James F. Oliviero, III, President, Chief Executive Officer and Director 
               |  |  |  |  | 994,665 |  |  |  |  |  | 4,774,392 |  |  |  |  |  | 2,765,264 |  |  |  |  |  | 13,273,267 |  |  |  |  |  | 18,047,659 |  |  | 
| 
                William Garrett Gray, Chief Financial Officer, Corporate Secretary and Treasurer 
               |  |  |  |  | 532,897 |  |  |  |  |  | 2,557,906 |  |  |  |  |  | 913,425 |  |  |  |  |  | 4,384,440 |  |  |  |  |  | 6,942,346 |  |  | 
| Directors |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  |  | 
| 
                Michael S. Weiss, Chairman of the Checkpoint Board 
               |  |  |  |  | 70,517 |  |  |  |  |  | 338,482 |  |  |  |  |  | 104,295 |  |  |  |  |  | 500,616 |  |  |  |  |  | 839,098 |  |  | 
| 
                Christian Béchon, Director 
               |  |  |  |  | 25,228 |  |  |  |  |  | 121,094 |  |  |  |  |  | 104,295 |  |  |  |  |  | 500,616 |  |  |  |  |  | 621,710 |  |  | 
| 
                Neil Herskowitz, Director 
               |  |  |  |  | 30,517 |  |  |  |  |  | 146,482 |  |  |  |  |  | 104,295 |  |  |  |  |  | 500,616 |  |  |  |  |  | 647,098 |  |  | 
| 
                Lindsay A. Rosenwald, M.D. 
               |  |  |  |  | 90,517 |  |  |  |  |  | 434,482 |  |  |  |  |  | 104,295 |  |  |  |  |  | 500,616 |  |  |  |  |  | 935,098 |  |  | 
| 
                Barry Salzman, Director 
               |  |  |  |  | 30,517 |  |  |  |  |  | 146,482 |  |  |  |  |  | 104,295 |  |  |  |  |  | 500,616 |  |  |  |  |  | 647,098 |  |  | 
| 
                Amit Sharma, M.D., Director 
               |  |  |  |  | — |  |  |  |  |  | — |  |  |  |  |  | 82,051 |  |  |  |  |  | 393,845 |  |  |  |  |  | 393,845 |  |  | 
|  |  |  | 
                Common Stock Beneficially Owned 
               |  | |||||||||
| 
                Name and Address of Beneficial Owner(1)
               |  |  | 
                Amount and
                 Nature of Beneficial Ownership |  |  | 
                Percentage of
                 Total Common Stock |  | ||||||
| 
                Michael S. Weiss 
               |  |  |  |  | 174,812(2) |  |  |  |  |  | 0.2%(2) |  |  | 
| 
                James F. Oliviero 
               |  |  |  |  | 3,759,929 |  |  |  |  |  | 4.4% |  |  | 
| 
                William Garrett Gray 
               |  |  |  |  | 1,446,322 |  |  |  |  |  | 1.7% |  |  | 
| 
                Lindsay A. Rosenwald, M.D. 
               |  |  |  |  | 194,812(2) |  |  |  |  |  | 0.2%(2) |  |  | 
| 
                Neil Herskowitz 
               |  |  |  |  | 134,812 |  |  |  |  |  | 0.2% |  |  | 
| 
                Christian Béchon 
               |  |  |  |  | 129,523 |  |  |  |  |  | 0.2% |  |  | 
| 
                Barry Salzman 
               |  |  |  |  | 134,812 |  |  |  |  |  | 0.2% |  |  | 
| 
                Amit Sharma, M.D. 
               |  |  |  |  | 82,051 |  |  |  |  |  | 0.1% |  |  | 
| 
                All executive officers and directors as a group 
               |  |  |  |  | 5,957,073(3) |  |  |  |  |  | 6.9%(3) |  |  | 
| 5% or Greater Stockholders: |  |  |  |  |  |  |  |  |  |  |  |  |  | 
| 
                Fortress Biotech, Inc. 
               |  |  |  |  | 6,222,249(4) |  |  |  |  |  | 7.2% |  |  | 
| 
                Beryl Capital Management LLC 
               |  |  |  |  | 6,074,216(5) |  |  |  |  |  | 7.0% |  |  | 
| 
                Armistice Capital, LLC 
               |  |  |  |  | 5,216,445(6) |  |  |  |  |  | 6.0% |  |  | 
|  |  |  | 
                Class A Common Stock
                 Beneficially Owned |  | |||||||||
| 
                Name and Address of Beneficial Owner 
               |  |  | 
                Amount and
                 Nature of Beneficial Ownership |  |  | 
                Percentage of
                 Total Class A Common Stock |  | ||||||
| 
                Fortress Biotech, Inc. 
               |  |  |  |  | 700,000 |  |  |  |  |  | 100% |  |  | 
|  |  |  | 
                Common Stock Beneficially Owned Assuming
                 Conversion of Class A Common Stock to Common Stock |  | |||||||||
| 
                Name and Address of Beneficial Owner 
               |  |  | 
                Amount and
                 Nature of Beneficial Ownership |  |  | 
                Percentage of
                 Total Common Stock |  | ||||||
| 
                Fortress Biotech, Inc. 
               |  |  |  |  | 6,922,249(1) |  |  |  |  |  | 8.0%(2) |  |  | 
|  |  |  | 
                Page 
               |  | |||
|  |  |  |  | A-1-2 |  |  | |
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|  |  |  |  |  |  |  |  | 
![[MISSING IMAGE: lg_locustwalk-4c.jpg]](lg_locustwalk-4c.jpg) 
        |  | 
                /s/ Andy Meyerson
                
                Locust Walk Securities LLC
               |  |  |  |  | 
![[MISSING IMAGE: lg_kroll-4c.jpg]](lg_kroll-4c.jpg) 
        ![[MISSING IMAGE: ft_kroll-4c.jpg]](ft_kroll-4c.jpg) 
        |  | 
                /s/ Duff & Phelps
                |  |  | ||
|  | Duff & Phelps Opinions Practice Kroll, LLC |  |  |  |  | 
![[MISSING IMAGE: px_25checkpointannual01-bw.jpg]](px_25checkpointannual01-bw.jpg) 
        ![[MISSING IMAGE: px_25checkpointannual02-bw.jpg]](px_25checkpointannual02-bw.jpg)